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Onye na-emepụta ntụ ntụ Amino Tadalafil Nọmba CAS: 385769-84-6 98% ịdị ọcha nkeji maka ihe mgbakwunye

Nkọwa Dị Mkpirikpi:

Amino Tadalafil bụ ihe mejupụtara ya yiri Tadalafil, ebe ụfọdụ otu ọrụ dị na nhazi ya ka amino otu nọchiri anya ya.


Nkọwa Ngwaahịa

Akara Ngwaahịa

Vidiyo Ngwaahịa

Usoro Ngwaahịa

Aha ngwaahịa

Amino Tadalafil

Aha ọzọ

(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A-Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dion e;(6R,12aR)-2-Amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4(6H,7H)-dione

Nọmba CAS

385769-84-6

Usoro molekụla

C21H18N4O4

Ibu molekụla

390.39

Ịdị ọcha

98.0%

Ọdịdị

Ntụ ntụ ọcha ruo na ntụ ọcha na-acha ọcha

Ngwa

Ihe Mgbakwunye Nri Ihe Ndị A Na-anaghị Ewu

Okwu mmeghe ngwaahịa

Amino Tadalafil bụ ihe ọhụrụ, ihe sitere na tadalafil, nke na-aghọwanye ewu ewu n'ọhịa nke nsogbu erectile (ED). Ọ na-ejikọta amino acid na tadalafil, ihe mgbochi PDE5 nke FDA kwadoro nke a na-ejikarị agwọ ED. Ọ na-arụ ọrụ site n'ịbawanye ọbara na amụ, na-enye ụmụ nwoke ohere iru ma nọgide na-enwe ahụ ike. Amino acid, n'aka nke ọzọ, na-arụ ọrụ dị mkpa na ọrụ dị iche iche nke ahụ, gụnyere mmepụta nke protein, nke bụ ihe owuwu nke anụ ahụ na akụkụ ahụ. A na-eme njikọta nke ihe abụọ a iji mee ka arụmọrụ Tadalafil dịkwuo mma n'ịgwọ ED. Amino Tadalafil bụkwa ụdị emelitere nke nwere ike pụrụ iche, na-eme ka arụmọrụ na ịdị iche iche nke onye bu ya ụzọ dịkwuo mma. Ọdịdị kemịkalụ ya ka dị ka Tadalafil, mana site na iwebata otu amino, ọ na-enweta àgwà pụrụ iche nke na-eme ka ọ pụta ìhè n'ụwa ọgwụ. Dị ka tadalafil, Amino Tadalafil na-arụ ọrụ site na igbochi phosphodiesterase 5 (PDE5), enzyme nke na-akpata imebi cyclic guanosine monophosphate (cGMP) n'ahụ. cGMP bụ ihe e kere eke nke na-akwalite izu ike nke arịa ọbara, si otú a na-eme ka ọbara na-erugharị nke ọma. Site na igbochi PDE5, amino Tadalafil na-eme ka cGMP na-agbakọta, si otú a na-eme ka vasodilation dịkwuo mma ma na-eme ka ọbara na-agbagharị nke ọma. Na mgbakwunye, ndị nchọpụta enyochaala ike ya iji nyere aka gwọọ benign prostatic hyperplasia (BPH) site n'ịkwalite ọbara na prostate.

atụmatụ

(1) Ịdị ọcha dị elu: Amino Tadalafil nwere ike inweta ngwaahịa dị ọcha dị elu site na usoro mmepụta dị mma. Ịdị ọcha dị elu pụtara nnweta bioavail ka mma na obere mmeghachi omume ọjọọ.

(2)Nchekwa: Nchekwa dị elu, obere mmeghachi omume ọjọọ.

(3) Ịkwụsi Ike: Amino Tadalafil nwere ezigbo nkwụsi ike ma nwee ike ịnọgide na-arụ ọrụ na mmetụta ya n'okpuru gburugburu ebe obibi na ọnọdụ nchekwa dị iche iche.

Ngwa

Amino Tadalafil bụ ihe na-egbochi PDE5 nke nwere otu mmetụta ọgwụ dịka tadalafil. Site na ijikọta amino acid na tadalafil, a na-eche na amino Tadalafil dị irè karịa n'ịgwọ ọrịa erectile karịa tadalafil naanị. Amino acid nwere ike inyere aka mee ka ọbara gbasaa ma kwado arụmọrụ zuru oke nke ọgwụ. Na mgbakwunye, ọ nwere ike ime ka mgbaàmà nke nsogbu erectile (ED) ka mma site na igbochi ọrụ nke enzyme PDE5 iji kwalite ọbara na-eruba n'ahụ ụmụ nwoke. Ma e jiri ya tụnyere tadalafil, amino Tadalafil na-agbanwe nwayọ nwayọ n'ime ahụ ma nwee ike imepụta mmetụta na-adịgide adịgide. Nke a na-enye amino Tadalafil nnukwu ikike n'ịgwọ ED.


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