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Fasoracetam ntụ ntụ CAS Nọmba: 110958-19-5 99% ịdị ọcha nkeji maka ihe mgbakwunye

Nkọwa Dị Mkpirikpi:

Ọgwụ kemịkalụ Fasoracetam bụ ọgwụ sịntetik nke otu ọgwụ a na-akpọ dihydropyridine pyrrolidone.


Nkọwa Ngwaahịa

Akara Ngwaahịa

Vidiyo Ngwaahịa

Usoro Ngwaahịa

Aha ngwaahịa

Fasoracetam

Aha ọzọ

FOSORACETAM;

(5R)-5-(piperidine-1-carbonyl)-2-pyrrolidone;

(5R)-5-(piperidine-1-carbonyl)pyrrolidin-2-one;

(5R)-5-piperidin-1-ylcarbonylpyrrolidin-2-otu

Nọmba CAS

110958-19-5

Usoro molekụla

C10H16N2O2

Ibu molekụla

196.25

Ịdị ọcha

99.0%

Ọdịdị

Ntụ ntụ ọcha

Nkwakọ ngwaahịa

1 kg/akpa 25kg/drum

Ngwa

Nootropic

Okwu mmeghe ngwaahịa

Fasoracetam, bụ ihe mejupụtara nootropic nke e mepụtara na Japan. Ọ na-ejikọta ihe ndị yiri ya na ndị ọzọ na-agba ọsọ dịka piracetam, mana ọ na-egosipụta njirimara pụrụ iche nke ihe omume. A na-eche na Fasoracetam na-agbanwe mmetụta nke ọtụtụ neurotransmitters n'ụbụrụ, gụnyere GABA, glutamatergic, na cholinergic sistem. Site na imetụta ntọhapụ na nnabata nke neurotransmitters ndị a, fasoracetam nwere ike imeziwanye ọrụ nghọta dịka nlebara anya, njikọta ebe nchekwa, na nhazi ozi. Nnyocha na ihe akaebe akụkọ na-egosi na fasoracetam nwere ike inye ọtụtụ uru nghọta. Otu n'ime ihe ndị bụ isi ya bụ ime ka ntinye uche na oge nlebara anya dịkwuo mma, na-eme ka ọ bụrụ onye enyemaka nwere ike inye aka maka ndị na-arịa nsogbu enweghị nlebara anya ma ọ bụ nsogbu enweghị nlebara anya (ADD/ADHD). Ọmụmụ ihe mbụ egosila nsonaazụ dị mma, na-egosi ikike fasoracetam imeziwanye nlebara anya, belata ihe ndọghachi azụ ma melite njikwa nghọta. Na mgbakwunye, ọmụmụ anụmanụ na-egosi na Fasoracetam na-eme ka ike ogologo oge dịkwuo mma, usoro metụtara nhazi ebe nchekwa na plasticity synaptic.

atụmatụ

(1) Ịdị ọcha dị elu: Fasoracetam nwere ike inweta ngwaahịa dị ọcha dị elu site na usoro mmepụta dị mma. Ịdị ọcha dị elu pụtara nnweta bioavailability ka mma na obere mmeghachi omume ọjọọ.

(2) Nchekwa: Ọmụmụ ihe egosila na a na-anabata fasoracetam nke ọma, ọ naghịkwa enwe mmetụta dị ukwuu mgbe ejiri ya mee ihe n'ime ọgwụ akwadoro.

(3) Ịkwụsi ike: Fasoracetam nwere ezigbo nkwụsi ike ma nwee ike ịnọgide na-arụ ọrụ na mmetụta ya n'okpuru gburugburu ebe obibi na ọnọdụ nchekwa dị iche iche.

Ngwa

Fasoracetam apụtala dị ka ihe na-adọrọ mmasị nke nwere ike ime ka ikike nghọta dịkwuo mma, ọkachasị ebe nchekwa, nlebara anya, na mmụta, a pụkwara iji ya mee ihe dị ka ihe mgbakwunye nri. Ngwaahịa a na-arụ ọrụ dị ka ihe na-eme ka ncheta dịkwuo mma site n'ịkpalite ndị na-anabata glutamate metabolic. N'ọhịa bayoloji, a na-ejikwa Fasoracetam dị ka ihe na-egbochi nhọrọ iji mụọ usoro bayoloji dị ka ihe ngosi mkpụrụ ndụ na apoptosis.


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