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Onye na-emepụta ntụ ntụ Coluracetam Nọmba CAS: 135463-81-9 99% ọcha nkeji maka ihe mgbakwunye

Nkọwa Dị Mkpirikpi:

Coluracetam bụ otu n'ime ezinụlọ racetam nke ihe ndị na-adịghị arụ ọrụ nke ọma, a makwaara ya dị ka MKC-231. Ụlọ ọrụ Kobe Pharmaceutical dị na Japan mepụtara ya iji gwọọ AD na nsogbu ọgụgụ isi.


Nkọwa Ngwaahịa

Akara Ngwaahịa

Vidiyo Ngwaahịa

Usoro Ngwaahịa

Aha ngwaahịa

Coluracetam

Aha ọzọ

MKC-231;

2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl)-1-pyrrolidineacetamide

Nọmba CAS

135463-81-9

Usoro molekụla

C19H23N3O3

Ibu molekụla

341.4

Ịdị ọcha

99.0%

Ọdịdị

Ntụ ntụ ọcha

Ngwa

Ihe Mgbakwunye Nri Ihe Ndị A Na-anaghị Ewu

Okwu mmeghe ngwaahịa

Coluracetam, onye otu ezinụlọ ndị otu agbụrụ nke ogige nootropic, nke a makwaara dị ka MKC-231, bụ ihe mejupụtara nootropic nke nwere mmụba nghọta na mmetụta neuroprotective. Coluracetam na-arụ ọrụ site na ịgbanwe usoro cholinergic. A na-eche na ọ na-eme ka ọkwa acetylcholine dịkwuo elu, isi ihe na-akpata neurotransmitter n'ụbụrụ nke jikọtara ya na mmụta na ọrụ ncheta. Coluracetam na-eme nke a site n'ịbawanye ọnụọgụ na ọrụ nke ndị na-ebuga choline, si otú a na-eme ka ntọhapụ nke acetylcholine dịkwuo mma ma na-eme ka akara ngosi dị n'etiti neurons dịkwuo mma. Ụfọdụ ọmụmụ nnwale na anụmanụ mbụ na-atụ aro na Coluracetam nwere ike inwe mmetụta neuroprotective na cognition-uplication. Ụfọdụ ọmụmụ ihe ndị ọzọ achọpụtala na Coluracetam nwere mmetụta mmezi ụfọdụ na nsogbu ncheta na ụdị AD.

atụmatụ

(1) Ịdị ọcha dị elu: A na-eji usoro mwepụ na mmepụta dị elu kwadebe Coluracetam iji hụ na ịdị ọcha dị elu. Ịdị ọcha dị elu a na-enyere aka imeziwanye nnweta bioavailability ma belata ihe omume nke mmeghachi omume ọjọọ.
(2) Nchekwa: A na-ewere Coluracetam dị ka ihe dị mma maka mmadụ. Ọtụtụ nnyocha egosila na ọ nwere obere nsí na obere mmetụta ọjọọ n'ime oke ọgwụ akwadoro.
(3) Ịkwụsi Ike: Nkwadebe Coluracetam na-egosipụta nkwụsi ike dị mma ma nwee ike ịnọgide na-arụ ọrụ na arụmọrụ ha n'okpuru gburugburu ebe obibi na ọnọdụ nchekwa dị iche iche. Nkwụsi ike a na-eme ka arụmọrụ kwụsiri ike ma bụrụ nke a pụrụ ịtụkwasị obi ruo ogologo oge.

Ngwa

A na-eji Coluracetam eme ihe ugbu a n'ọtụtụ ụzọ dị iche iche ma na-egosi nkwa dị mma n'ọdịnihu. A na-ejikarị ya eme ihe dị ka ihe mgbakwunye nri na-eme ka ọgụgụ isi dịkwuo mma, ndị mmadụ na-achọkwa ime ka ebe nchekwa, itinye uche, na mmụta dịkwuo mma. A na-eche na ikike nke ngwakọta ahụ iji gbanwee usoro cholinergic na-enyere aka na mmetụta ya na-eme ka nghọta dịkwuo mma. Na mgbakwunye, nnyocha na-egosi na Coluracetam nwere ike inwe ihe nchebe neuroprotective nke nwere ike inye aka gbochie mbelata ọgụgụ isi nke afọ ma na-akwado ahụike ụbụrụ zuru oke.


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