Noopept(GVS-111) onye na-emepụta ntụ ntụ CAS Nọmba: 157115-85-0 99% ịdị ọcha nkeji maka ihe mgbakwunye
Usoro Ngwaahịa
| Aha ngwaahịa | Noopept,GVS-111 |
| Aha ọzọ | N-(1-(Phenylacetyl)-L-prolyl)glycine ethyl ester |
| Nọmba CAS | 157115-85-0 |
| Usoro molekụla | C17H22N2O4 |
| Ibu molekụla | 318.37 |
| Ịdị ọcha | 99.5% |
| Ọdịdị | ntụ ntụ ọcha |
| Nkwakọ ngwaahịa | 25kg/mgbịrịgba |
| Ngwa | nootropics |
Okwu mmeghe ngwaahịa
Noopept bụ ngwakọta peptide sịntetik e mepụtara na Russia na 1990s iji melite ọrụ nghọta. A na-ekewa ya dị ka nootropic, nke pụtara na ọ na-eme ka arụmọrụ ụbụrụ na ikike nghọta dịkwuo mma, gụnyere ebe nchekwa, itinye uche, na mmụta. Noopept na-eme ka ebe nchekwa na mmụta dịkwuo mma site n'ịkwalite ntọhapụ nke ụfọdụ neurotransmitters nke na-akpali ọrụ neuron. Nke a na-enyere aka ịmepụta ncheta ọhụrụ ma chekwaa ozi nke ọma. Na mgbakwunye, a na-eche na Noopept nwere mmetụta dị mma na ntinye uche zuru oke. Site n'ịkwalite echiche doro anya, ọ na-eme ka mmepụta na arụmọrụ dịkwuo mma n'ọtụtụ ọrụ, ma ọ bụ ịmụ ma ọ bụ ịrụ ọrụ na ọrụ dị mgbagwoju anya. Nnyocha ndị metụtara ya na-egosi na Noopept nwere ike inwe ihe nchebe neuroprotective megide nrụgide oxidative na neurotoxicity. A na-eche na ihe ndị a na-enyere aka igbochi mbelata nghọta metụtara afọ ma belata ihe egwu nke ọrịa neurodegenerative.
atụmatụ
(1) Ịdị ọcha dị elu: Noopept nwere ike inweta ngwaahịa dị ọcha dị elu site na usoro mmepụta dị mma. Ịdị ọcha dị elu pụtara nnweta bioavailability ka mma na obere mmeghachi omume ọjọọ.
(2) Nchekwa: A chọpụtala na Noopept dị mma maka ahụ mmadụ.
(3) Ịkwụsi Ike: Noopept nwere ezigbo nkwụsi ike ma nwee ike ịnọgide na-arụ ọrụ na mmetụta ya n'okpuru gburugburu ebe obibi na ọnọdụ nchekwa dị iche iche.
Ngwa
Dịka ihe mgbakwunye nri, Noopept na-eme ka nguzozi dị n'etiti sistemụ akwara na sistemụ antioxidant dịkwuo mma, na-agbanwe ọrụ dị iche iche nke ahụ, gụnyere nghọta na nchekasị, ma na-eme ka ebe nchekwa dịkwuo mma n'ọtụtụ ọnọdụ. Iri Noopept ogologo oge nwere ike inye aka mee ka ọkwa nke ihe na-eto eto akwara (NGF) na ihe na-akpata neurotrophic (BDNF) nke ụbụrụ pụta, ọkachasị na mpaghara ụbụrụ dịka hippocampus na hypothalamus. Noopept nwere ike inwe mmetụta ụfọdụ na ọrụ GABA na hippocampus, usoro ụbụrụ nke a na-echekarị na ọ na-etinye aka na ncheta. A gosikwara na Noopept na-achịkwa usoro acetylcholine na ụbụrụ. Iweghachi nkwekọ dị n'etiti ọrụ glutamate na acetylcholine abụghị naanị na-echebe ụbụrụ gị pụọ na mmebi. Ọ nwere ike ime ka nghọta, ncheta, mmụta, icheta, ọnọdụ, na ibelata nchekasị.












