Galantamine Hydrobromide ntụ ntụ emeputa CAS No.: 1953-04-4 98% ịdị ọcha min.maka ihe mgbakwunye
Ngwa ngwaahịa
Aha ngwaahịa | Galantamine hydrobromide |
Aha ọzọ | Galanthamine hydrobromide; Galantamine HBr; Galanthamine HBr; (4aS,6R,8aS) -4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-6H-Benzofuro[3a,3,2-ef] [2] benzazepin- 6-ol, Hydrobromide |
CAS Mba. | 1953-04-4 |
Usoro ihe omimi | C17H21NO3.HBr |
Ibu molekụla | 368.27 |
Ịdị ọcha | 98.0% |
Ọdịdị | na-acha ọcha na-acha ọcha ntụ ntụ |
Nkwakọ ngwaahịa | 1kg / akpa 10kgs,25kgs /drum |
Ngwa | nootropics |
Ntinye ngwaahịa
Galantamine hydrobromide bụ ụdị benzozepine sitere na bulbs na ifuru nke narcissus, osmanthus, ma ọ bụ canna.Ọ bụkwa ihe mgbochi cholinesterase nke ọnụ.Dị ka njikọ nke nicotinic acetylcholine receptor, ejirila ya mee ihe iji kwalite ọrụ neurocognitive.Ọrụ ya bụ ịsọ mpi na ngbanwe na-egbochi acetylcholinesterase, si otú ahụ na-abawanye mkpokọta acetylcholine.
Mgbe etinyere ya n'ọbara, galanthamine hydrobromide na-abanye ngwa ngwa n'akụkụ niile nke ahụ, gụnyere ụbụrụ.Ọ na-ejikọta na nicotinic acetylcholine receptor, na-eme mgbanwe mgbanwe na mmụba acetylcholine ntọhapụ.Ọ na-arụkwa ọrụ site na ịsọ mpi na ịtụgharị mmetụta nke ndị na-egbochi cholinesterase.Site na igbochi cholinesterase, ọ na-egbochi ire ere nke acetylcholine, si otú a na-abawanye ọkwa na ogologo oge nke neurotransmitter dị ike.Galanthamine na-emekwa ka mmụta na ikike ncheta dịkwuo mma, na-egbochi mbufụt ụbụrụ ma na-edobe ọkwa dị elu nke neurotransmitters site n'ịkwado iguzosi ike n'ezi ihe nke neurons na synapses.
Njirimara
(1) Mmetụta ọzọ bara uru nke galanthamine hydrobromide na nkwalite ebe nchekwa bụ ikike ya ịkwalite ọrụ ebe nchekwa.Ọ na-abawanye ọsọ nke nhazi ebe nchekwa ma mee ka njigide nkọwa na eziokwu dịkwuo mma.
(2) A na-eme ka ikike mmụta dịkwuo mma site na ịba ụba synaptic plasticity na neuroplasticity.Galanthamine hydrobromide na-emetụta neuroplasticity ozugbo ma ọ bụ na-apụtaghị ìhè.Ọ na-akpali plastik synapti site na ịgbalite microglia na astrocyte.
(3) Ọ na-enyere aka ihi ụra ma na-amụba izu ike.Galanthamine nwere ike ime ka ihe isi ike nke ọnọdụ ihi ụra dịkwuo elu site n'ịkpalite ụra anya ngwa ngwa ngwa ngwa, si otú a na-eme ka ụra dịkwuo mma.
(4) Mee ka nchebe antioxidant dịkwuo mma, Galantamine na-enye nchebe antioxidant iji lụso nrụgide oxidative kpatara site na free radicals.Ọ nwere ike ichebe mkpụrụ ndụ ụbụrụ site na mmebi oxidative iji nọgide na-arụ ọrụ ụbụrụ kacha mma.