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Tianeptine Semisulfate Monohydrate ntụ ntụ emeputa CAS No .: 1224690-84-9 98% ịdị ọcha min.maka ihe mgbakwunye

Nkọwa dị mkpirikpi:

Tianeptine Hemisulfate Monohydrate bụ onye na-emechi ihe nchịkwa serotonin nke ahọpụtara (SSRI) yana ọgwụ na-egbochi ịda mbà n'obi.


Nkọwa ngwaahịa

Mkpado ngwaahịa

Ngwa ngwaahịa

Aha ngwaahịa

Tianeptine Hemisulfate Monohydrate

Aha ọzọ

tianeptinesulfate;

(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;

7-[(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f] [1,2] thiazepin-11-yl) amino] heptanoicacidsulfatehydrate (2: 1: 2);

Tianeptinehemisulfatemonohydrate (THM);

7-[(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f] [1,2] thiazepin-11-yl) amino] heptanoicacidsulfatehydrate (2: 1: 2);

Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;

THM

CAS Mba.

1224690-84-9

Usoro ihe omimi

C21H27ClN2O8S2

Ibu molekụla

535.02

Ịdị ọcha

98.0%

Ọdịdị

kristal ọcha ntụ ntụ

Ngwa

Ihe mgbakwunye nri nri

Ntinye ngwaahịa

Tianeptine Hemisulfate Monohydrate bụ onye na-emechi ihe nchịkwa serotonin nke ahọpụtara (SSRI) yana ọgwụ na-egbochi ịda mbà n'obi.Dị ka ihe na-abụghị omenala antidepressant, usoro ya dị iche na nke omenala antidepressants, na-eme ka ọnọdụ na mmetụta uche dịkwuo mma site n'ịkwalite plasticity synaptic nke neurons hippocampal.A na-ejikwa Tianeptine Hemisulfate Monohydrate agwọ nchekasị na nsogbu ọnọdụ uche.

A na-eji Tianeptine Hemisulfate Monohydrate mee ihe n'ọtụtụ ebe na nyocha ahụike, ọkachasị na mmepe nke antidepressants.A na-enyochakwa ya maka iji ya na ọrịa neurodegenerative, nchịkwa mgbu, na ọgwụgwọ riri ahụ.A na-enyocha arụmọrụ nke Tianeptine Hemisulfate Monohydrate n'ọtụtụ ebe ma kwadoro ya, a kwadoro ya maka ọgwụgwọ ịda mbà n'obi n'ọtụtụ mba.

Ekwesiri iburu n'uche na ebe Tianeptine Hemisulfate Monohydrate egosila na ọ bụ ihe na-egbochi ịda mbà n'obi na ngwa ngwa ụlọ ọgwụ, a na-ekewa ya dị ka ihe a na-achịkwa na mba ụfọdụ, na-egbochi iji ya na ire ere.Onye ọ bụla na-eji ma ọ bụ na-azụta Tianeptine Hemisulfate Monohydrate kwesịrị ịma iwu na ụkpụrụ dị mkpa na obodo ha.

Njirimara

(1) Usoro pụrụ iche nke ime ihe: Tianeptine Hemisulfate Monohydrate bụ ihe na-eme ka serotonin reuptake enhancer (SSRE), nke pụtara na ọ na-eme ka nchịkọta nke serotonin dị n'ụbụrụ, na-eduga na ụba synaptic plasticity na mma ọnọdụ.Usoro omume a dị iche na antidepressants ọdịnala, nke na-abụkarị ndị inhibitors reuptake serotonin (SSRIs).
(2) Nmalite ngwa ngwa: Tianeptine Hemisulfate Monohydrate na-eme ngwa ngwa na-arụ ọrụ ngwa ngwa, na ọmụmụ ụlọ ọgwụ na-egosi ọganihu na mgbaàmà ịda mbà n'obi dị ka otu izu mgbe mmalite ọgwụgwọ gasịrị.
(3) Ọrụ ọgụgụ isi na-emeziwanye: Tianeptine Hemisulfate Monohydrate egosipụtara iji meziwanye ọrụ ọgụgụ isi na ndị ọrịa nwere nnukwu nsogbu ịda mbà n'obi, dị ka ebe nchekwa na nlebara anya.

(4) Ike riri ahụ dị ala: N'adịghị ka antidepressants ndị ọzọ, Tianeptine Hemisulfate Monohydrate nwere ikike iri ahụ dị ala ma ọ naghị akpata mgbagha mgbagha mgbe a kwụsịrị.Nke a bụ n'ihi na ọ naghị elekwasị anya na usoro dopamine, nke jikọtara ya na ịṅụ ọgwụ ọjọọ na ịdabere na ya.

(5) Ọgwụgwọ nsogbu nchekasị: Tianeptine Hemisulfate Monohydrate egosila na ọ nwere mmetụta anxiolytic, na-eme ka ọ bụrụ ọgwụgwọ nwere ike ime ka nsogbu nchekasị dị ka nsogbu nchekasị zuru oke na nchekasị mmekọrịta ọha na eze.

Ngwa

Tianeptine Hemisulfate Monohydrate bụ kemịkalụ ọgwụ a na-ejikarị eme ihe na ngalaba ụlọ ọgwụ na nyocha.Dị ka ọgwụ na-egbochi ịda mbà n'obi, a kwadoro ya n'ọtụtụ mba maka ọgwụgwọ ịda mbà n'obi, nchekasị, nsogbu ọnọdụ uche, na ọrịa ndị ọzọ metụtara ya.Na mgbakwunye, a mụọla Tianeptine Hemisulfate Monohydrate maka ike ya n'ịgwọ ọrịa neurodegenerative dị ka Alzheimer, njikwa mgbu, na ọgwụgwọ riri ahụ.

N'ime afọ ndị na-adịbeghị anya, Tianeptine Hemisulfate Monohydrate enwetawo mmụba na-ewu ewu na nyocha ahụike, karịsịa na mmepe nke ọgwụ ndị na-egbochi ịda mbà n'obi.N'ihe ọmụmụ ndị ọzọ na-akwado mmetụta ọgwụgwọ ya, atụmanya ntinye ya na-eji nwayọọ nwayọọ pụta ìhè.Tianeptine Hemisulfate Monohydrate nwere ike ịghọ ọgwụ na-arụ ọrụ dị iche iche maka ịgwọ ọrịa dị iche iche nke akwara ozi n'ọdịnihu.

Ọzọkwa, Tianeptine Hemisulfate Monohydrate nwekwara ike ngwa na ubi ndị ọzọ.Nnyocha e mere n'oge na-adịbeghị anya gosiri na Tianeptine Hemisulfate Monohydrate nwere ike ịnwe ike ịgwọ ọrịa ọrịa neurofunctional post-stroke.Na mgbakwunye, ụfọdụ ọmụmụ na-atụ aro na Tianeptine Hemisulfate Monohydrate nwere ike ịba uru maka ọrịa metabolic dị ka oke ibu na ọrịa shuga.


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