J-147 onye na-emepụta ntụ ntụ CAS No.: 1146963-51-0 99.0% ịdị ọcha min.maka ihe mgbakwunye
Ngwa ngwaahịa
Aha ngwaahịa | 2,2,2-Trifluoroacetic acid 1- (2,4-DiMethylphenyl) -2-[(3-Methoxyphenyl) Methylene] hydrazide] |
Aha ọzọ | J-147, J147 |
CAS Mba. | 1146963-51-0 |
Usoro ihe omimi | C18H17F3N2O2 |
Ibu molekụla | 350.33 |
Ịdị ọcha | 99% |
Ọdịdị | Ọcha ntụ ntụ |
Nkwakọ ngwaahịa | 1kg kwa akpa |
Ngwa | nootropics |
Okwu Mmalite ngwaahịa
J-147 bụ neuroprotectant na-arụ ọrụ nke ọma nke sitere na curcumin, ihe na-arụ ọrụ na turmeric.N'adịghị ka curcumin, ọ na-agafe ihe mgbochi ụbụrụ ọbara nke ọma.N'ime ha, J-147 na-arụ ọrụ site na ijikọ ATP synthase.Mmepụta nke ATP na-ejikọta ya na usoro ịka nká.Na mgbakwunye na ịbawanye ọkwa nke neurotransmitters NGF na BDNF, J-147 nwere ike ịchịkwa nke a.Na mgbakwunye, J-147 na-egbochi monoamine oxidase B na dopamine transporter.Na-akwalite uto ụbụrụ site n'ịbawanye ọkwa nke ihe na-eto eto (NGF) na ụbụrụ neurotrophic factor (BDNF).Nke kachasị mkpa, J-147 nwere ike ịkwalite uto nke mkpụrụ ndụ akwara ọhụrụ, kwalite ikike mmụta na ebe nchekwa ụbụrụ, ma melite ọrụ ọgụgụ isi.
Njirimara
(1) Ịdị ọcha dị elu: J-147 nwere ike nweta ngwaahịa dị ọcha site na nhazi usoro mmepụta ihe.Ịdị ọcha dị elu pụtara bioavailability ka mma yana mmeghachi omume ọjọọ dị ole na ole.
(2) Nchekwa: J-147 egosila na ọ dị mma maka ahụ mmadụ.
(3) Nkwụsi ike: J-147 nwere ezigbo nkwụsi ike ma nwee ike ịnọgide na-arụ ọrụ ya na mmetụta ya n'okpuru ebe dị iche iche na ọnọdụ nchekwa.
(4) Ọ dị mfe itinye uche: J-147 nwere ike ịbanye ngwa ngwa site na ahụ mmadụ, na-abanye n'ọbara ọbara site na eriri afọ, kesaa ya na anụ ahụ na akụkụ dị iche iche.
Ngwa
J-147 bụ ihe sịntetik nke usoro izizi ya gụnyere nkwalite mitochondrial, si otú a na-ebuli mmepụta ike na ọkwa cellular.Emebere J-147 iji kwalite ikike ụbụrụ imezi yana chebe onwe ya pụọ na mmebi metụtara afọ site na imeziwanye ọrụ mitochondrial.Na mgbakwunye, J-147 na-egosipụta ihe mgbochi mkpali na ihe antioxidant, na-eme ka mmetụta neuroprotective ya dịkwuo elu.J-147 nwere ike ịkwalite uto nke mkpụrụ ndụ akwara ọhụrụ, kwalite ikike mmụta na ebe nchekwa ụbụrụ, ma melite ọrụ ọgụgụ isi.