YDL223C (HBT1) onye na-emepụta ntụ ntụ CAS No.: 489408-02-8 99% ịdị ọcha min.maka ihe mgbakwunye
Ngwa ngwaahịa
Aha ngwaahịa | HBT1 |
Aha ọzọ | YDL223C |
CAS Mba. | 489408-02-8 |
Usoro ihe omimi | C16H17F3N4O2S |
Ibu molekụla | 386.40 |
Ịdị ọcha | 99.0% |
Ọdịdị | Agba odo siri ike |
Nkwakọ ngwaahịa | 1kg kwa akpa 25kg kwa drum |
Ngwa | nootropics |
Ntinye ngwaahịa
HBT1 na-ejikọta na ngalaba njikọ njikọ nke α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor (AMPA-R) n'ụzọ dabere na glutamate.Nke a pụtara na HBT1 bụ molekul nwere ike jikọta naanị na saịtị akọwapụtara na protein AMPA-R mgbe glutamate dị, yana njikọ a na-enyere aka ịhazi ọrụ protein.A na-egosipụta ndị na-anabata AMPA n'ime usoro nhụjuanya etiti ma na-arụ ọrụ dị mkpa na nkwurịta okwu neuronal, nhazi mmetụta, na mmụta, ebe nchekwa, na synapti plasticity.Ndị na-anabata AMPA bụ ndị na-enye aka na neurotransmission na-akpali akpali, na-agba ọsọ ngwa ngwa, ngwa ngwa enweghị mmasị nke ọtụtụ synapses, ma na-etinye aka na nzaghachi mbụ nke mpaghara synapti na glutamate.A na-ejikọta ndị na-anabata AMPA na ndị na-anabata NMDA na synapses, na ọnụ ha na-akwalite usoro synaptic plasticity gụnyere mmụta, ebe nchekwa, excitotoxicity, na neuroprotection.
Njirimara
Ihe na-akpata ụbụrụ ụbụrụ (BDNF) bụ ihe na-akpata neurotrophic nke na-arụ ọrụ dị mkpa na nhazi na mgbasawanye nke neurons, ma nwee mmetụta dị ike na ọtụtụ mmetụta na mmụba, ọdịiche, nlanarị na ọnwụ nke mkpụrụ ndụ neuronal na ndị na-abụghị neuronal, Ọrụ dị ka a neurotransmitter modulator na-enye aka na neuronal plasticity maka mmụta na ebe nchekwa.Ya mere, ọ dị mkpa maka ahụike na ọdịmma nke usoro ụjọ ahụ.Mmụba na BDNF nwere ike inye aka na ọgwụgwọ na mgbochi nke ọtụtụ ọrịa.
Ngwa
HBT1 bụ ihe nkwalite ihe nnabata AMPA nke nwere obere mgbu ma e jiri ya tụnyere LY451395 na OXP1, ọ na-ebute mmepụta nke ụbụrụ neurotrophic nke sitere na ụbụrụ (BDNF), ọ na-egosikwa ntakịrị mmetụta na mgbakasị neurons mbụ.HBT1 na-ejikọta na ngalaba njikọ njikọ nke AMPA-R n'ụzọ dabere na glutamate.Ọnụ, ha na-akwalite usoro synaptic plasticity nke gụnyere mmụta, ebe nchekwa, excitability na neuroprotection.Ọ nwere ike melite ikike ọgụgụ isi na ebe nchekwa nke ụbụrụ, ma kwalite ikike mmụta ndị mmadụ.