Amino Tadalafil ntụ ntụ emeputa CAS No.: 385769-84-6 98% ịdị ọcha min. maka ihe mgbakwunye
Video ngwaahịa
Ngwa ngwaahịa
Aha ngwaahịa | Amino Tadalafil |
Aha ọzọ | (6R,12aR) -2-Amino-6- (1,3-benzodioxol-5-yl) -2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b] indole-1,4-dione; AminoTadalafil (6R,12Ar) -2-Amino-6-(1,3-Benzodioxol-5-Yl) -2,3,6,7,12,12A -Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR) -2-Amino-6-(benzo[d] [1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R) ,12aR) -2-amino-6- (benzo [d][1,3]dioxol-5-yl) -2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3] ,4-b]indole-1,4(6H,7H)-dione |
CAS Mba. | 385769-84-6 |
Usoro ihe omimi | C21H18N4O4 |
Ibu arọ molekụla | 390.39 |
Ịdị ọcha | 98.0% |
Ọdịdị | Na-acha ọcha na-acha ọcha ntụ ntụ |
Ngwa | Ihe mgbakwunye nri nri |
Ntinye ngwaahịa
Amino Tadalafil bụ ihe ọhụrụ dị ọhụrụ, nke sitere na tadalafil, nke na-aghọwanye ewu ewu n'ọhịa nke nrụrụ erectile (ED). Ọ na-ejikọta amino acid na tadalafil, ihe mgbochi PDE5 nke FDA kwadoro nke a na-ejikarị emeso ED. Ọ na-arụ ọrụ site n'ịbawanye ọbara na-eruba na amụ, na-enye ohere ka ụmụ nwoke nweta ma nọgide na-arụ ọrụ. N'aka nke ọzọ, amino acid na-ekere òkè dị mkpa n'ọrụ dị iche iche nke ahụ, gụnyere mmepụta nke protein, nke bụ ihe na-ewulite anụ ahụ na akụkụ ahụ. Ejikọtara ngwakọta nke ihe abụọ a iji mee ka Tadalafil dị irè n'ịgwọ ED. Na amino Tadalafil bụ ụdị emelitere nke nwere ikike pụrụ iche, na-eme ka arụmọrụ na ike dị iche iche nke onye bu ya ụzọ pụta. Ọdịdị kemịkal ya ka dị ka Tadalafil, ma site na ntinye nke amino dị iche iche, ọ na-enweta àgwà pụrụ iche nke na-eme ka ọ pụta ìhè na ụwa ọgwụ. Dị ka tadalafil, Amino Tadalafil na-arụ ọrụ site na igbochi phosphodiesterase 5 (PDE5), enzyme na-ahụ maka ịkụda cyclic guanosine monophosphate (cGMP) n'ime ahụ. cGMP bụ ihe okike nke na-akwalite izu ike nke arịa ọbara, si otú ahụ na-abawanye mmụba ọbara. Site na igbochi PDE5, amino Tadalafil na-eme ka nchịkọta nke cGMP dị elu, si otú a na-eme ka vasodilation dịkwuo mma ma na-eme ka mgbasa ọbara dịkwuo mma. Na mgbakwunye, ndị nchọpụta enyochala ikike ọ nwere inye aka na-agwọ ọrịa hyperplasia prostate na-adịghị mma (BPH) site n'ịkwalite ịgbasa ọbara na prostate.
Njirimara
(1) Ịdị ọcha dị elu: Amino Tadalafil nwere ike nweta ngwaahịa dị ọcha site na nhazi usoro mmepụta ihe. Ịdị ọcha dị elu pụtara bioavailability ka mma yana mmeghachi omume ọjọọ dị ole na ole.
(2) Nchekwa: Nchekwa dị elu, mmeghachi omume ọjọọ ole na ole.
(3) Nkwụsi ike: Amino Tadalafil nwere ezigbo nkwụsi ike ma nwee ike ịnọgide na-arụ ọrụ ya na mmetụta ya n'okpuru ebe dị iche iche na ọnọdụ nchekwa.
Ngwa
Amino Tadalafil bụ onye na-emechi PDE5 nwere otu mmetụta ọgwụ dị ka tadalafil. Site na ijikọta amino acid na tadalafil, a na-eche na amino Tadalafil dị irè karị n'ịgwọ ọrịa erectile karịa tadalafil naanị. Amino acid nwere ike inye aka kwalite mgbasa ọbara ma kwado ịdị irè nke ọgwụ n'ozuzu ya. Tụkwasị na nke ahụ, ọ nwere ike imeziwanye ihe mgbaàmà nke nrụrụ erectile (ED) site na igbochi ọrụ nke enzyme PDE5 iji kwalite ọbara na-eruba na akụkụ ọmụmụ nwoke. N'iji ya tụnyere tadalafil, amino Tadalafil na-eji nwayọọ nwayọọ na-emegharị n'ime ahụ ma nwee ike ịmepụta mmetụta na-adịte aka. Nke a na-enye amino Tadalafil ikike dị ukwuu n'ịgwọ ED.