Nefiracetam ntụ ntụ emeputa CAS No .: 77191-36-7 99% ịdị ọcha min. maka ihe mgbakwunye
Video ngwaahịa
Ngwa ngwaahịa
| Aha ngwaahịa | Nefiracetam |
| Aha ọzọ | n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamide; NEFIRACETAM; 2-oxo-1-pyrrolidinylaceticacid,2,6-dimethylanilide; dm9384; n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamid; DM-9384, (2- (2-Oxopyrrolidin-1-yl) -N- (2,6-dimethylphenyl) -acetamide; DMPA |
| CAS Mba. | 77191-36-7 |
| Usoro ihe omimi | C14H18N2O2 |
| Ibu arọ molekụla | 246.3 |
| Ịdị ọcha | 99.0% |
| Ọdịdị | Ọcha ntụ ntụ |
| Nkwakọ ngwaahịa | 25 n'arọ / gbọmgbọm |
| Ngwa | nootropic |
Ntinye ngwaahịa
Nefiracetam bụ nke ezinụlọ piracetam, otu ọgwụ ndị a maara maka ihe ndị na-eme ka ha nwee mmetụta. Nefiracetam bụ nke mbụ synthesized na mmalite 1980 na ngwa ngwa dọtara uche n'ihi na ya pụrụ iche usoro nke edinam na ike ọgwụgwọ ngwa. A na-eche na ogige agbụrụ a na-emetụta neurotransmitters na ndị na-anabata ya na ụbụrụ, n'ikpeazụ na-akwalite ikike ọgụgụ isi ka mma. Nefiracetam na-emetụta ụbụrụ ụbụrụ acetylcholine, isi ihe na-ahụ maka ebe nchekwa, mmụta, na ọrụ ọgụgụ isi. Site n'ịgbanwe ndị na-anabata acetylcholine, nefiracetam na-akwalite mgbasawanye nkwurịta okwu n'etiti neurons, si otú ahụ na-eme ka synaptic plasticity dịkwuo mma ma na-eme ka nchekwa nchekwa dịkwuo mma. Na mgbakwunye, nefiracetam na-emekọ ihe na ndị na-anabata gamma-aminobutyric acid (GABA) iji nyere aka dozie milieu neurotransmitter. Site n'imetụta ndị na-eme ihe na-akpali akpali na ndị na-emechi emechi, nefiracetam na-enyere aka ịnọgide na-arụ ọrụ ụbụrụ kachasị mma, si otú ahụ na-eme ka elekwasị anya, nlebara anya, na ịrụ ọrụ n'ozuzu ya.
Njirimara
(1) Ịdị ọcha dị elu: Nefiracetam nwere ike nweta ngwaahịa dị ọcha site na ịmecha usoro mmepụta ihe. Ịdị ọcha dị elu pụtara bioavailability ka mma yana mmeghachi omume ọjọọ dị ole na ole.
(2) Nchekwa: Nchekwa dị elu, mmeghachi omume ọjọọ ole na ole.
(3) Nkwụsi ike: Nefiracetam nwere nkwụsi ike dị mma ma nwee ike ịnọgide na-arụ ọrụ ya na mmetụta ya n'okpuru ebe dị iche iche na ọnọdụ nchekwa.
Ngwa
Nefiracetam bụ ihe mgbapụta hydrophobic nke piracetam, nke a na-ewerekarị dị ka ihe na-ahụ maka nchọpụta nke ọwa calcium n'ime ahụ na nnyefe na-apụtaghị ìhè nke ihe mgbaàmà na-akpali akpali dị ka onye na-eme ihe ike nke calcium ion channels. Ebe ejikọta Glycine nke NDMA nnata. Site na mmetụta ya na ụbụrụ ụbụrụ ụbụrụ, nefiracetam nwere ike ịkwalite ikike ọgụgụ isi ma gbochie mmụta na nsogbu ncheta. Ọ nweghị muscarinic agonist receptor agonist ma ọ bụ ihe na-emegide ya, ọ dịghịkwa egbochi ọrụ acetylcholinease. Ya mere, a na-enweta mmetụta mgbochi-mnestic na ebe nchekwa ya site n'ịkwalite ntọhapụ nke acetylcholine na cortex cerebral.
