PRL-8-53 onye na-emepụta ntụ ntụ CAS No .: 51352-87-5 98% ịdị ọcha min. maka ihe mgbakwunye
Ngwa ngwaahịa
| Aha ngwaahịa | PRL-8-53 |
| Aha ọzọ | Methyl 3- (2- (benzyl (Methyl) amino) ethyl) benzoate hydrochloride; benzoic acid, 3-[2-[methyl (phenylmethyl) amino] ethyl] -, methyl ester, hydrochloride (1: 1) ; Methyl 3- {2-[benzyl (methyl) amino] ethyl} benzoate hydrochloride (1: 1) |
| CAS Mba. | 51352-87-5 |
| Usoro ihe omimi | C18H22ClNO2 |
| Ibu arọ molekụla | 319.83 |
| Ịdị ọcha | 98.0% |
| Ọdịdị | Ọcha ntụ ntụ |
| Nkwakọ ngwaahịa | 1 n'arọ kwa akpa 25kg / drum |
| Ngwa | nootropic |
Ntinye ngwaahịa
PRL-8-53, nke a makwaara dị ka methyl 3- (2- (benzyl (methyl) amino) ethyl) benzoate, bụ ngwakọta nootropic sịntetik nke a na-eche iji kwalite nnyefe cholinergic ma na-achịkwa ọkwa dopamine na ụbụrụ. Àgwà ndị a na-enye aka na mmetụta ya nwere ike ime ka ọgụgụ isi dịkwuo elu, si otú ahụ na-eme ka nhazi ebe nchekwa dịkwuo mma, njide, na iweghachite. Ọtụtụ nchọpụta banyere anụmanụ na ụmụ mmadụ akọpụtala ihe dị mma maka ihe ndị na-eme ka ncheta ya dịkwuo mma. N'ime nyocha abụọ nke kpuru ìsì, nchọpụta pilot na-achịkwa placebo, isiokwu ndị natara otu dose nke PRL-8-53 gosipụtara ikike nchekwa okwu ka mma na ikike iweghachite ma e jiri ya tụnyere otu placebo. Nchọpụta ndị a kpalitere mmasị na nyocha ndị ọzọ gbasara ikike ogige ahụ. Nnyocha ọzọ n'ime oke gosiri na inye PRL-8-53 mere ka ikike ha mụta ihe n'ọrụ mmiri. Oke ndị ejiri PRL-8-53 emeso ya nwere ike ịchọta ikpo okwu zoro ezo nke ọma karịa njikwa, na-egosipụta ikike nke ogige ahụ dị ka nkwalite ebe nchekwa.
Njirimara
(1) Ịdị ọcha dị elu: PRL-8-53 nwere ike nweta ngwaahịa dị ọcha site na nhazi usoro mmepụta ihe. Ịdị ọcha dị elu pụtara bioavailability ka mma yana mmeghachi omume ọjọọ dị ole na ole.
(2) Nchekwa: Nchekwa dị elu, mmeghachi omume ọjọọ ole na ole, enweghị mmeghachi omume ọjọọ doro anya.
(3) Nkwụsi ike: PRL-8-53 nwere ezigbo nkwụsi ike ma nwee ike ịnọgide na-arụ ọrụ ya na mmetụta ya n'okpuru ebe dị iche iche na ọnọdụ nchekwa.
Ngwa
Dị ka ụdị mgbakwunye nkwalite nkwalite ọhụụ ọhụrụ, PRL-8-53 na-eme ka ebe nchekwa dị mkpụmkpụ na ebe nchekwa na-arụ ọrụ dịkwuo mma, ebe ọ na-eme ka ikike mmụta na ọsọ nweta nka, na-enyere aka melite mmụta na ịrụ ọrụ nke ọma. Nnyocha na-egosi na PRL-8-53 nwere ike ịkwalite uto na mmeghari nke neurons na ụbụrụ. PRL-8-53 nwere ike ịbawanye ọsọ nke ụbụrụ na-ahazi ozi, na-enye ndị mmadụ ohere ịrụzu ọrụ na ime mkpebi ngwa ngwa. Ọ bụ ezie na e jiri ya tụnyere ogige nootropic ndị ọzọ Otú ọ dị, nchọpụta na PRL-8-53 dị oke, ma nchọpụta dị adị na-egosi na ọ nwere ike imeziwanye ebe nchekwa na ikike ọgụgụ isi.
